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Dr Martin J Scanlon
Senior Lecturer
BSc University of Leeds (UK)
PhD University of Nottingham (UK)
Phone: +61 3 9903 9540
Fax: +61 3 9903 9582
Email: martin.scanlon@pharm.monash.edu.au
Medicinal Chemistry and Drug Action, Monash Institute of Pharmaceutical Sciences
- Fragment-based drug design
- Structure-based design of novel anti-microbial agents
- Analysis of protein-ligand interactions
- Protein structure determination and structural biology
Education
- Spectrometric identification of small molecules
- Drug-protein interactions
Representative publications
- Velkov T, Lim, ML, Horne J, Simpson JS, Porter CJ, Scanlon MJ. Characterization of lipophilic drug binding to rat intestinal fatty acid binding protein. Mol Cell Biochem. 2009 Jan 22. [Epub ahead of print].
- Heras B, Shouldice SR, Totsika M, Scanlon MJ, Schembri MA, Martin JL. DSB proteins and bacterial pathogenicity. Nat Rev Microbiol. 2009;7:215-225.
- Vivian JP, Scoullar J, Robertson AL, Bottomley SP, Horne J, Chin Y, et.al. Structural and biochemical characterization of the oxidoreductase NmDsbA3 from Neisseria meningitidis. J Biol Chem. 2008; 283:32452-32461.
- Robertson AL, Horne J, Ellisdon AM, Thomas B, Scanlon MJ, Bottomley SP. The structural impact of a polyglutamine tract is location-dependent. Biophys J. 2008; 95:5922-5930.
- Roberts BP, Scanlon MJ, Krippner GY, Chalmers DK. The Dotted Cap Notation: A Concise Notation for Describing Variegated Dendrimers. New J Chem 2008; 32,:1543-1554.
- Headey SJ, Vom A, Simpson JS, Scanlon MJ. Backbone assignments of the 34 kDa ketopantoate reductase from E. coli. Biomol NMR Assignments. 2008; 2:93-96.
- Chuang S, Velkov T, Horne J, Porter CJ, Scanlon MJ. Characterization of the drug binding specificity of rat liver fatty acid binding protein. J Med Chem. 2008; 51:3755-3764.
- Velkov T, Horne J, Laguerre A, Jones E, Scanlon MJ, and Peter CJ.Examination of the role of intestinal Fatty Acid-binding protein in drug absorption using a parallel artificial membrane permeability assay. Chem Biol. 2007; 14:453-465.
- Horne J, Scanlon MJ. Backbone and side chain 1H, 15N and 13C assignments for the reduced form of the oxidoreductase protein DsbA from Vibrio cholerae. Biomol NMR Assignments 2007; 1:75-76.
- Horne J, d'Auvergne EJ, Coles M, Velkov T, Chin, Y, Charman WN, et.al. Probing the flexibility of the DsbA oxidoreductase from Vibrio cholerae--a 15N - 1H heteronuclear NMR relaxation analysis of oxidized and reduced forms of DsbA. J Mol Biol. 2007; 371:703-716.
- Perry CS, Charman SA, Prankerd RJ, Chiu FC, Scanlon MJ, Chalmers D, et.al. The binding interaction of synthetic ozonide antimalarials with natural and modified beta-cyclodextrins. J Pharm Sci. 2006; 95:146-158.
- Gibbs GM, Scanlon MJ, Swarbrick J, Curtis S, Gallant E, Dulhunty AF, et.al. The cysteine-rich secretory protein domain of Tpx-1 is related to ion channel toxins and regulates ryanodine receptor Ca2+ signaling. J Biol Chem. 2006; 281:4156-4163.
- Velkov T, Chuang S, Wielens J, Sakellaris H, Charman WN, Peter CJ et.al. The interaction of lipophilic drugs with intestinal fatty acid-binding protein. J Biol Chem. 2005; 280:17769-17776.
- Velkov T, Chuang S, Prankerd R, Sakellaris H, Peter CJ, Scanlon MJ. An improved method for the purification of rat liver-type fatty acid binding protein from Escherichia coli. Protein Expr Purif. 2005; 44:23-31.
- Jennings CV, Rosengren KJ, Daly NL, Plan M, Stevens J, Scanlon MJ, et.al. Isolation, Solution Structure, and Insecticidal Activity of Kalata B2, a Circular Protein with a Twist: Do Mobius Strips Exist in Nature? Biochemistry. 2005; 44:851-860.
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